Tag agonist [67 articles] Export

Recent papers classified by the tag agonist.

	Ligand-regulated oligomerization of beta(2)-adrenoceptors in a model lipid bilayer. [My Copy] The EMBO journal (17 September 2009) by Juan José J. Fung, Xavier Deupi, Leonardo Pardo, et al.Xiao Jie J. Yao, Gisselle A. Velez-Ruiz, Brian T. Devree, Roger K. Sunahara, Brian K. Kobilka posted to oligomerization inverse_agonist fret b2ar antagonist agonist by xdeupi on 2009-10-06 19:26:56 as
	Exploring the mechanism of agonist efficacy: a relationship between efficacy and agonist dissociation rate at the muscarinic M3 receptor. [My Copy] Molecular pharmacology, Vol. 76, No. 3. (September 2009), pp. 543-551. by David A. Sykes, Mark R. Dowling, Steven J. Charlton posted to efficacy drug binding_kinetics binding agonist by xdeupi on 2009-10-06 17:50:31 as
	Hot-Spots-Guided Receptor-Based Pharmacophores (HS-Pharm): A Knowledge-Based Approach to Identify Ligand-Anchoring Atoms in Protein Cavities and Prioritize Structure-Based Pharmacophores [My Copy] Journal of Chemical Information and Modeling, Vol. 48, No. 7. (1 July 2008), pp. 1396-1410. by Caterina Barillari, Gilles Marcou, Didier Rognan posted to theory pharmacology ligands drug docking binding b2ar agonist by xdeupi on 2009-10-05 18:45:05 as along with 3 people tbinbal superpyrin higueruelo
	Dopamine Controls Persistence of Long-Term Memory Storage ドーパミンが長期記憶の貯蔵の持続性を調節している [My Copy] Science, Vol. 325, No. 5943. (21 August 2009), pp. 1017-1020. by Janine I. Rossato, Lia R. M. Bevilaqua, Ivan Izquierdo, Jorge H. Medina, Martin Cammarota posted to vta ventral tegmental receptor rat memory ltm long-term hippocampus dorsal dopamine d1 area antagonist agonist by ttaga on 2009-08-31 08:33:02 as along with 5 people tyrell_turing davidcsterratt fpbattaglia PaperCollector ckemere
	Conserved and sexually dimorphic behavioral responses to biogenic amines in decapitated Drosophila [My Copy] Proceedings of the National Academy of Sciences of the United States of America, Vol. 94, No. 8. (15 April 1997), pp. 4131-4136. by Chris Yellman, Heng Tao, Biao He, Jay Hirsh posted to sex receptor drosophila dopamine d2receptor d1receptor behavior antagonist amine agonist by bangyuzhou on 2009-08-25 08:19:20 as
	Small-molecule agonists for the thyrotropin receptor stimulate thyroid function in human thyrocytes and mice. [My Copy] Proceedings of the National Academy of Sciences of the United States of America (10 July 2009) by Susanne Neumann, Wenwei Huang, Steve Titus, et al.Gerd Krause, Gunnar Kleinau, Anna Teresa T. Alberobello, Wei Zheng, Noel T. Southall, James Inglese, Christopher P. Austin, Francesco S. Celi, Oksana Gavrilova, Craig J. Thomas, Bruce M. Raaka, Marvin C. Gershengorn posted to agonist gpcr gphr ligand small tmd tshr by gcaltabiano on 2009-07-21 08:10:25 as
	Allosteric modulation of muscarinic acetylcholine receptors. [My Copy] Current neuropharmacology, Vol. 5, No. 3. (September 2007), pp. 157-167. by K. J. Gregory, P. M. Sexton, A. Christopoulos posted to activation agonist binding kinetics ligands pharmacology by xdeupi on 2009-07-20 18:21:37 as
	Suppression of excitatory cholinergic synaptic transmission by Drosophila dopamine D1-like receptors [My Copy] European Journal of Neuroscience, Vol. 26, No. 9. (November 2007), pp. 2417-2427. by Ning Yuan, Daewoo Lee posted to receptor drosophila dopamine d1receptor antagonist agonist by bangyuzhou on 2009-05-22 03:10:17 as
	A membrane-based microfluidic device for controlling the flux of platelet agonists into flowing blood. [My Copy] Lab on a chip, Vol. 8, No. 5. (May 2008), pp. 701-709. by K. B. Neeves, S. L. Diamond posted to agonist convection microfluidics platelet by matthewhflamm on 2009-05-18 19:33:12 as
	Sequence-Derived Three-Dimensional Pharmacophore Models for G-Protein-Coupled Receptors and Their Application in Virtual Screening [My Copy] Journal of Medicinal Chemistry, Vol. 0, No. 0. (0000) by Thomas Klabunde, Clemens Giegerich, Andreas Evers posted to agonist antagonist binding drug ligands modeling pharmacology by xdeupi on 2009-05-06 09:59:59 as along with 1 person reyez
	Conformational toggle switches implicated in basal constitutive and agonist-induced activated states of 5-hydroxytryptamine-4 receptors. [My Copy] Molecular pharmacology, Vol. 75, No. 4. (April 2009), pp. 982-990. by L. P. Pellissier, J. Sallander, M. Campillo, et al.F. Gaven, E. Queffeulou, M. Pillot, A. Dumuis, S. Claeysen, J. Bockaert, L. Pardo posted to activation agonist switch toggle by xdeupi on 2009-05-06 09:50:42 as along with 1 person arnaucordomi
	Identifying conformational changes of the β2 adrenoceptor that enable accurate prediction of ligand/receptor interactions and screening for GPCR modulators [My Copy] Journal of Computer-Aided Molecular Design by Kimberly Reynolds, Vsevolod Katritch, Ruben Abagyan posted to 2 adrenoceptor agonist gpcr homology ligand mmff model screening virtual by zimbo1 on 2009-04-15 16:16:04 as along with 1 person LamBras
	Triton x-100 inhibits AGonist-induced currents and suppresses benzodiazepine modulation of GABAA receptors in xenopus oocytes [My Copy] Biochimica et Biophysica Acta (BBA) - Biomembranes (12 February 2009) by Rikke Søgaard, Bjarke Ebert, Dan Klaerke, Thomas Werge posted to agonist amphipiles current gaba inhibit receptor sogaard09pdf by paulschlesinger on 2009-02-17 22:33:36 as
	Prediction of the 3D Structure and Dynamics of Human DP G-Protein Coupled Receptor Bound to an Agonist and an Antagonist [My Copy] J. Am. Chem. Soc., Vol. 129, No. 35. (5 September 2007), pp. 10720-10731. by Y. Li, F. Zhu, N. Vaidehi, et al.W. A. Goddard, F. Sheinerman, S. Reiling, I. Morize, L. Mu, K. Harris, A. Ardati, A. Laoui posted to agonist antagonist docking gpcr homologymodeling md moleculardynamics by sschurer on 2008-12-07 20:31:34 as along with 2 people daevans superpyrin
	Evaluation of an Estrogen Receptor-beta Agonist in Animal Models of Human Disease [My Copy] Endocrinology, Vol. 144, No. 10. (1 October 2003), pp. 4241-4249. by Heather A. Harris, Leo M. Albert, Yelena Leathurby, et al.Michael S. Malamas, Richard E. Mewshaw, Chris P. Miller, Yogendra P. Kharode, James Marzolf, Barry S. Komm, Richard C. Winneker, Donald E. Frail, Ruth A. Henderson, Yuan Zhu, James C. Keith posted to agonist animal-model beta estrogen-receptor by Zephyrus on 2008-11-19 13:50:12 as
	Fluorescent GPCR ligands as new tools in pharmacology. [My Copy] Current medicinal chemistry, Vol. 15, No. 21. (2008), pp. 2132-2143. by K. Kuder, K. Kieć-Kononowicz posted to activation agonist binding drug fluorescence imaging ligands by xdeupi on 2008-10-15 10:30:17 as
	Relationships Between Molecular Structure and Perceived Odor Quality of Ligands for a Human Olfactory Receptor [My Copy] Chem. Senses, Vol. 33, No. 7. (1 September 2008), pp. 639-653. by Guenhael Sanz, Thierry Thomas-Danguin, El H. Hamdani, et al.Claire Le Poupon, Loic Briand, Jean-Claude Pernollet, Elisabeth Guichard, Anne Tromelin posted to agonist code ligands or by serpar on 2008-09-28 04:39:39 as
	Ex vivo study of 5-HT(1A) and 5-HT(7) receptor agonists and antagonists on cAMP accumulation during memory formation and amnesia. [My Copy] Behavioural brain research (3 August 2008) by G Perez-García, A Meneses posted to 5-ht1a 5-ht7antagonist agonist antagonist memory by Fritz to the group neurolit on 2008-09-19 14:38:42 as
	Anesthesia for functional neurosurgery: the role of dexmedetomidine. [My Copy] Current opinion in anaesthesiology, Vol. 21, No. 5. (October 2008), pp. 537-543. by Irene Rozet posted to anesthesia dexmedetomidine neurosurgery agonist alpha-2-agonist by pmariana on 2008-09-12 16:14:40 as
	Recruitment of beta-arrestin2 to the dopamine D2 receptor: Insights into anti-psychotic and anti-parkinsonian drug receptor signaling. [My Copy] Neuropharmacology (8 April 2008) by Ib V V. Klewe, Søren M M. Nielsen, Louise Tarpø, et al.Eneko Urizar, Concetta Dipace, Jonathan A A. Javitch, Ulrik Gether, Jan Egebjerg, Kenneth V V. Christensen posted to activation active-state agonist arrestin biased_agonism binding disease fluorescence imaging internalization pharmacology by xdeupi on 2008-05-13 16:24:49 as
	Chemogenomic approaches to rational drug design [My Copy] Br J Pharmacol, Vol. 152, No. 1. (29 May 2007), pp. 38-52. by D. Rognan posted to agonist binding drug ligands pharmacology priviledged_structures by xdeupi to the group LabCompMed on 2008-03-28 15:54:47 as along with 4 people and 2 groups jmrivort jerome_ucsf_slb guhjy tjimenez G-quadruplex Supramolecular
	beta-Arrestin-biased Agonism at the beta2-Adrenergic Receptor. [My Copy] J Biol Chem, Vol. 283, No. 9. (29 February 2008), pp. 5669-5676. by M. T. Drake, J. D. Violin, E. J. Whalen, J. W. Wisler, S. K. Shenoy, R. J. Lefkowitz posted to activation agonist arrestin b2ar biased_agonism drug gproteins imaging internalization ligands pharmacology by xdeupi to the group LabCompMed on 2008-02-27 10:39:07 as
	Mechanisms of anti-inflammatory and neuroprotective actions of PPAR-gamma agonists. [My Copy] Front Biosci, Vol. 13 (2008), pp. 1813-1826. by R. Kapadia, J. H. Yi, R. Vemuganti posted to agonist antiinflammatorisch future ppar-gamma by viki on 2007-11-24 09:01:30 as
	[3H]Org 43553, the First Low Molecular Weight Agonistic and Allosteric Radioligand for the Human Luteinizing Hormone Receptor. [My Copy] Mol Pharmacol (7 November 2007) by Laura Heitman, Julia Oosterom, Kimberly Bonger, Cornelis Timmers, Peter Wiegerinck, Ad P P. Ijzerman posted to agonist hcg lhr lmw lowmolecularweigth by gcaltabiano on 2007-11-13 08:41:31 as
	Effects of CP-336,156, a New, Nonsteroidal Estrogen Agonist/Antagonist, on Bone, Serum Cholesterol, Uterus, and Body Composition in Rat Models [My Copy] Endocrinology, Vol. 139, No. 4. (1 April 1998), pp. 2068-2076. by Hua Z. Ke, Vishwas M. Paralkar, William A. Grasser, et al.Todd D. Crawford, Hong Qi, Hollis A. Simmons, Christine M. Pirie, Kristin L. Chidsey-Frink, Thomas A. Owen, Steven L. Smock, Hong K. Chen, Webster S. Jee, Kimberly O. Cameron, Robert L. Rosati, Thomas A. Brown, Paul Dasilva-Jardine, David D. Thompson posted to agonist antagonist body distribution estrogen fat rat by FW_Gibb on 2007-05-23 13:54:50 as
	Chromophore Channeling in the G-Protein Coupled Receptor Rhodopsin. [My Copy] J Am Chem Soc (15 May 2007) by Ting Wang, Yong Duan posted to rhodopsin modeling md ligands binding amber agonist activation by xdeupi to the group LabCompMed on 2007-05-21 10:04:04 as
	Multiple signaling states of G-protein-coupled receptors. [My Copy] Pharmacol Rev, Vol. 57, No. 2. (June 2005), pp. 147-161. by D. M. Perez, S. S. Karnik posted to activation agonist gpcr pharmacology review rhodopsin switch by xdeupi on 2007-04-26 14:57:25 as along with 1 group LabCompMed
	Role of group-conserved residues in the helical core of beta2-adrenergic receptor. [My Copy] Proc Natl Acad Sci U S A, Vol. 104, No. 17. (24 April 2007), pp. 7027-7032. by P. Chelikani, V. Hornak, M. Eilers, et al.P. J. Reeves, S. O. Smith, U. L. Rajbhandary, H. G. Khorana posted to tm4 switch ser b2ar agonist activation by xdeupi to the group LabCompMed on 2007-04-26 12:27:17 as
	"Phenotypic" pharmacology: the influence of cellular environment on G protein-coupled receptor antagonist and inverse agonist pharmacology. [My Copy] Biochem Pharmacol, Vol. 73, No. 6. (15 March 2007), pp. 737-751. by C. P. Nelson, R. A. Challiss posted to agonist gpcr ligands pharmacology by xdeupi on 2007-04-10 18:54:26 as along with 1 person and 2 groups Fritz neurolit LabCompMed
	Bioluminescence resonance energy transfer as a screening assay: Focus on partial and inverse agonism. [My Copy] J Biomol Screen, Vol. 12, No. 1. (February 2007), pp. 41-49. by L. Elster, C. Elling, A. Heding posted to ligands fret b2ar agonist activation by xdeupi to the group LabCompMed on 2007-04-10 18:50:15 as
	Real-time optical recording of beta1-adrenergic receptor activation reveals supersensitivity of the Arg389 variant to carvedilol. [My Copy] J Clin Invest, Vol. 117, No. 1. (January 2007), pp. 229-235. by F. Rochais, J. P. Vilardaga, V. O. Nikolaev, M. Bünemann, M. J. Lohse, S. Engelhardt posted to activation agonist b2ar helix8 mutation by xdeupi to the group LabCompMed on 2007-03-12 14:39:00 as
	Subclassification and nomenclature of alpha- and beta-adrenoceptors. [My Copy] Curr Top Med Chem, Vol. 7, No. 2. (2007), pp. 129-134. by J. P. Hieble posted to agonist b2ar drug genome ligands pharmacology review by xdeupi on 2007-03-12 14:33:19 as along with 1 group LabCompMed
	Recent advances in identification and characterization of beta-adrenoceptor agonists and antagonists. [My Copy] Curr Top Med Chem, Vol. 7, No. 2. (2007), pp. 207-216. by J. P. Hieble posted to agonist b2ar drug ligands pharmacology by xdeupi on 2007-03-12 14:32:04 as along with 1 group LabCompMed
	Effects of the potential 5-HT7 receptor agonist AS 19 in an autoshaping learning task. [My Copy] Behav Brain Res, Vol. 163, No. 1. (30 August 2005), pp. 136-140. by G. S. Perez-García, A. Meneses posted to 5-ht-receptors 5-ht7 agonist as19 by dark_innocent on 2007-02-14 13:30:09 as along with 1 person and 1 group Fritz neurolit
	Both Ligand- and Cell-Specific Parameters Control Ligand Agonism in a Kinetic Model of G Protein-Coupled Receptor Signaling. [My Copy] PLoS Comput Biol, Vol. 3, No. 1. (12 January 2007) by Tamara L L. Kinzer-Ursem, Jennifer J J. Linderman posted to activation agonist b2ar pharmacology by xdeupi to the group LabCompMed on 2007-02-13 15:38:17 as
	Identification of an agonist-induced conformational change occurring adjacent to the ligand-binding pocket of the M(3) muscarinic acetylcholine receptor. [My Copy] J Biol Chem, Vol. 280, No. 41. (14 October 2005), pp. 34849-34858. by S. J. Han, F. F. Hamdan, S. K. Kim, et al.K. A. Jacobson, L. M. Bloodworth, B. Li, J. Wess posted to ligands cation-pi binding agonist by xdeupi to the group LabCompMed on 2007-01-15 16:08:15 as
	Activation of the CXCR3 chemokine receptor through anchoring of a small molecule chelator ligand between TM-III, -IV and -VI. [My Copy] Mol Pharmacol (14 December 2006) by Mette M M. Rosenkilde, Michael B B. Andersen, Rie Nygaard, Thomas M M. Frimurer, Thue W W. Schwartz posted to ligands ionic chemokine cation-pi agonist activation by xdeupi to the group LabCompMed on 2007-01-11 16:06:35 as
	GluVII:06--a highly conserved and selective anchor point for non-peptide ligands in chemokine receptors. [My Copy] Curr Top Med Chem, Vol. 6, No. 13. (2006), pp. 1319-1333. by M. M. Rosenkilde, T. W. Schwartz posted to modeling ligands ionic chemokine binding agonist by xdeupi to the group LabCompMed on 2007-01-10 14:45:13 as
	Allosteric Activation of the Follicle-stimulating Hormone (FSH) Receptor by Selective, Nonpeptide Agonists [My Copy] J. Biol. Chem., Vol. 281, No. 19. (12 May 2006), pp. 13226-13233. by Stephen D. Yanofsky, Emily S. Shen, Frank Holden, et al.Erik Whitehorn, Barbara Aguilar, Emily Tate, Christopher P. Holmes, Randall Scheuerman, Derek Maclean, May M. Wu, Donald E. Frail, Francisco J. Lopez, Richard Winneker, Brian J. Arey, Ronald W. Barrett posted to agonist fsh by ndoelker to the group LabCompMed on 2006-11-07 14:52:10 as
	Movement of ‘gating charge’ is coupled to ligand binding in a G-protein-coupled receptor [My Copy] Nature (25 October 2006) by Yair Ben-Chaim, Baron Chanda, Nathan Dascal, Francisco Bezanilla, Itzchak Parnas, Hanna Parnas posted to activation agonist gpcr by cen4ik on 2006-11-02 13:03:34 as along with 1 person paulschlesinger
	Structure-affinity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agents. [My Copy] J Med Chem, Vol. 47, No. 26. (16 December 2004), pp. 6616-6624. by M. Leopoldo, F. Berardi, N. A. Colabufo, et al.M. Contino, E. Lacivita, M. Niso, R. Perrone, V. Tortorella posted to 5-ht7 agonist by Fritz on 2006-10-30 15:59:46 as along with 1 person and 1 group dark_innocent neurolit
	Choline is transported by vesicular acetylcholine transporter. [My Copy] J Neurochem, Vol. 91, No. 3. (November 2004), pp. 766-768. by D. T. Bravo, N. G. Kolmakova, S. M. Parsons posted to agonist choline receptor vacht by chenlc03 on 2006-10-11 12:26:31 as
	Novel mutants of the human beta1-adrenergic receptor reveal amino acids relevant for receptor activation. [My Copy] J Biol Chem, Vol. 281, No. 26. (30 June 2006), pp. 18120-18125. by B. Behr, C. Hoffmann, G. Ottolina, K. N. Klotz posted to activation agonist b2ar binding drug ligands modeling mutation pharmacology structure by xdeupi to the group LabCompMed on 2006-09-05 11:05:20 as
	Determining the Potency and Molecular Mechanism of Action of Insurmountable Antagonists. [My Copy] J Pharmacol Exp Ther (20 July 2006) by Terry P P. Kenakin, Stephen Jenkinson, Christian Watson posted to activation drug ligands agonist pharmacology by xdeupi to the group LabCompMed on 2006-09-05 09:51:58 as
	Glucose-lowering and insulin-sensitizing actions of exendin-4: studies in obese diabetic (ob/ob, db/db) mice, diabetic fatty Zucker rats, and diabetic rhesus monkeys (Macaca mulatta) [My Copy] Diabetes, Vol. 48, No. 5. (1 May 1999), pp. 1026-1034. by Aa Young, Br Gedulin, S. Bhavsar, et al.N. Bodkin, C. Jodka, B. Hansen, M. Denaro posted to 1 agonist biosci353 diabetes exenatide exendin-4 glp-1r glucagon like peptide by cherrie on 2006-08-04 03:49:13 as
	GPCR agonists and antagonists in the clinic. [My Copy] Med Chem, Vol. 1, No. 4. (July 2005), pp. 405-421. by J. D. Tyndall, R. Sandilya posted to agonist drug gpcr ligands pharmacology by xdeupi on 2006-07-24 10:18:01 as along with 1 group LabCompMed
	Data-Driven Analysis in Drug Discovery [My Copy] Journal of Receptors and Signal Transduction, Vol. 26, No. 4. (August 2006), pp. 299-327. by Terry Kenakin posted to agonist binding drug ligands pharmacology by xdeupi on 2006-07-17 16:28:05 as along with 1 group LabCompMed
	Molecular basis of inverse agonism in a G protein-coupled receptor. [My Copy] Nat Chem Biol, Vol. 1, No. 1. (June 2005), pp. 25-28. by J. P. Vilardaga, R. Steinmeyer, G. S. Harms, M. J. Lohse posted to agonist g-protein gpcr by Fritz to the group neurolit on 2006-07-07 22:12:21 as along with 1 person awooga
	Molecular evolution of adrenoceptors and dopamine receptors: implications for the binding of catecholamines. [My Copy] J Med Chem, Vol. 49, No. 5. (9 March 2006), pp. 1706-1719. by H. Xhaard, V. V. Rantanen, T. Nyrönen, M. S. Johnson posted to agonist b2ar binding gpcr ligands modeling by xdeupi on 2006-03-06 10:11:30 as along with 1 group LabCompMed
	Molecular mechanisms of beta2-adrenergic receptor function and regulation. [My Copy] Proc Am Thorac Soc, Vol. 2, No. 4. (2005) by D. W. McGraw, S. B. Liggett posted to activation agonist b2ar by xdeupi to the group LabCompMed on 2006-02-20 09:27:39 as

Note: You may cite this page as: http://www.citeulike.org/tag/agonist

Result page: 1 2 Next

activation	59
b2ar	46
ligands	39
binding	32
pharmacology	28
drug	22
gpcr	20
antagonist	15
ser	10
modeling	9
receptor	7
review	7
switch	7
rhodopsin	6
5-ht7	5
memory	5
5-ht1a	4
5-ht7antagonist	4
cation-pi	4
channel	4
chemokine	4
fluorescence	4
imaging	4
ionic	4
mutation	4
tm5	4
arrestin	3
biased_agonism	3
dopamine	3
fret	3
internalization	3
md	3
p2x	3
toggle	3
5-ht-receptors	2
amber	2
as19	2
auta08_neuph_55_148	2
behavior	2
calcium	2
cardiac	2
ccr5	2
d1receptor	2
docking	2
drosophila	2
ecl2	2
fpl64176	2
fsh	2
g-protein	2
gabaa	2
genome	2
gproteins	2
helix	2
helix8	2
histamine	2
ligand	2
loops	2
lp44	2
n745	2
npxxy	2
pdf	2
priviledged_structures	2
rat	2
s542	2
structure	2
subtype	2
tm4	2
tm6	2
transmembrane	2
adrenoceptor	1
aggression	1
amphipiles	1
beta	1
biting	1
body	1
code	1
current	1
dexmedetomidine	1
efficacy	1
events	1
exenatide	1
exendin-4	1
gaba	1
glp-1r	1
gphr	1
hcg	1
inverse_agonist	1
kinetics	1
lowmolecularweigth	1
ltcc	1
moleculardynamics	1
oligomerization	1
or	1
release	1
small	1
sogaard09pdf	1
tegmental	1
theory	1
tmd	1
virtual	1

Tag agonist [67 articles] Export

Related Tags