patricia's library 90 articles Export

	The structure and function of G-protein-coupled receptors [My Copy] Nature, Vol. 459, No. 7245. (20 May 2009), pp. 356-363. by Daniel M. Rosenbaum, Soren G. F. Rasmussen, Brian K. Kobilka posted to function gpcr review structure by patricia on 2009-06-10 17:23:25 as along with 8 people diod guhjy viktor21614 agrossfield xdeupi akundaje hsekiguc barry
	Nonallergic angioedema: role of bradykinin [My Copy] Allergy, Vol. 62, No. 8. (August 2007), pp. 842-856. by Bas, M., Adams, et al. V., Suvorava, T., Niehues, T., Hoffmann, T. K., Kojda, G. posted to bradykinin pharmacology by patricia on 2007-08-31 09:42:58 as
	B-9972 is an inactivation-resistant agonist of the bradykinin B2 receptor derived from the peptide antagonist B-9430: pharmacologic profile and effective induction of receptor degradation. [My Copy] J Pharmacol Exp Ther (15 August 2007) by Marie-Therese T. Bawolak, Lajos Gera, Guillaume Morissette, John M M. Stewart, Francois Marceau posted to analogues b2 by patricia on 2007-08-31 09:28:14 as
	Constitutive activation of the alpha 1B-adrenergic receptor by all amino acid substitutions at a single site. Evidence for a region which constrains receptor activation. [My Copy] J Biol Chem, Vol. 267, No. 3. (25 January 1992), pp. 1430-1433. by M. A. Kjelsberg, S. Cotecchia, J. Ostrowski, M. G. Caron, R. J. Lefkowitz posted to activation general gpcr by patricia on 2007-05-14 11:21:34 as
	Novel series of O-substituted 8-quinolines and 4-benzothiazoles as potent antagonists of the bradykinin B2 receptors. [My Copy] Bioorg Med Chem Lett, Vol. 9, No. 3. (8 February 1999), pp. 327-332. by H. Heitsch, A. Wagner, B. A. Schölkens, K. Wirth posted to antagonist b2 bradykinin by patricia on 2007-03-14 12:14:30 as
	Bradykinin B2 receptor as a potential therapeutic target. [My Copy] Drug News Perspect, Vol. 13, No. 4. (May 2000), pp. 213-225. by H. Heitsch posted to b2 pharmacology receptor by patricia on 2007-03-14 12:11:59 as
	Na+ ions binding to the bradykinin B2 receptor suppress agonist-independent receptor activation. [My Copy] Biochemistry, Vol. 35, No. 41. (15 October 1996), pp. 13368-13377. by U. Quitterer, S. AbdAlla, K. Jarnagin, W. Müller-Esterl posted to b2 bradykinin mutation receptor by patricia on 2007-03-02 15:45:35 as
	Identification of a ligand-dependent switch within a muscarinic receptor. [My Copy] J Biol Chem, Vol. 273, No. 34. (21 August 1998), pp. 21563-21568. by T. A. Spalding, E. S. Burstein, S. C. Henderson, K. R. Ducote, M. R. Brann posted to activation gpcr receptor by patricia on 2007-03-02 13:20:40 as
	Effect of different treatments of long-range interactions and sampling conditions in molecular dynamic simulations of rhodopsin embedded in a dipalmitoyl phosphatidylcholine bilayer. [My Copy] J Comput Chem (31 January 2007) by Arnau Cordomí, Olle Edholm, Juan J J. Perez posted to gpcr receptor by patricia on 2007-03-02 12:24:05 as along with 2 people and 1 group xdeupi arnaucordomi LabCompMed
	Critical role of electrostatic interactions of amino acids at the cytoplasmic region of helices 3 and 6 in rhodopsin conformational properties and activation. [My Copy] J Biol Chem (23 February 2007) by Eva Ramon, Arnau Cordomi, Laia Bosch, et al.Evgeni Yu Y. Zernii, Ivan I I. Senin, Joan Manyosa, Pavel P P. Philippov, Juan J J. Perez, Pere Garriga posted to gpcr receptor by patricia on 2007-03-02 12:02:14 as along with 1 person arnaucordomi
	Biomolecular modeling: Goals, problems, perspectives. [My Copy] Angewandte Chemie (International ed. in English), Vol. 45, No. 25. (19 June 2006), pp. 4064-4092. by Wilfred F. van Gunsteren, Dirk Bakowies, Riccardo Baron, et al.Indira Chandrasekhar, Markus Christen, Xavier Daura, Peter Gee, Daan P. Geerke, Alice Glättli, Philippe H. Hünenberger, Mika A. Kastenholz, Chris Oostenbrink, Merijn Schenk, Daniel Trzesniak, Nico F. van der Vegt, Haibo B. Yu posted to md modeling review by patricia on 2007-02-23 11:33:08 as along with 2 people mijogiffin LamBras
	G-protein-coupled receptors and cancer [My Copy] Nature Reviews Cancer, Vol. 7, No. 2., pp. 79-94. by Robert T. Dorsam, Silvio J. Gutkind posted to cancer gpcr by patricia on 2007-02-23 09:56:25 as
	Nonpeptide ligands that target peptide-activated GPCRs in inflammation. [My Copy] Curr Med Chem, Vol. 12, No. 25. (2005), pp. 3027-3042. by J. S. Blakeney, D. P. Fairlie posted to antagonist gpcr inflammation by patricia on 2007-02-22 11:52:52 as
	Bradykinin B1 antagonists: SAR studies in the 2,3-diaminopyridine series. [My Copy] Bioorg Med Chem Lett, Vol. 15, No. 17. (1 September 2005), pp. 3925-3929. by S. D. Kuduk, R. K. Chang, C. Ng, et al.K. L. Murphy, R. W. Ransom, C. Tang, T. Prueksaritanont, R. M. Freidinger, D. J. Pettibone, M. G. Bock posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:47:57 as
	2,3-Diaminopyridine as a platform for designing structurally unique nonpeptide bradykinin B1 receptor antagonists. [My Copy] Bioorg Med Chem Lett, Vol. 15, No. 9. (2 May 2005), pp. 2385-2388. by D. M. Feng, J. M. Wai, S. D. Kuduk, et al.C. Ng, K. L. Murphy, R. W. Ransom, D. Reiss, R. S. Chang, C. M. Harrell, T. MacNeil, C. Tang, T. Prueksaritanont, R. M. Freidinger, D. J. Pettibone, M. G. Bock posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:45:05 as
	5-Piperazinyl pyridine carboxamide bradykinin B1 antagonists. [My Copy] Bioorg Med Chem Lett, Vol. 16, No. 10. (15 May 2006), pp. 2791-2795. by S. D. Kuduk, C. N. Di Marco, R. K. Chang, et al.M. R. Wood, J. J. Kim, K. M. Schirripa, K. L. Murphy, R. W. Ransom, C. Tang, M. Torrent, S. Ha, T. Prueksaritanont, D. J. Pettibone, M. G. Bock posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:38:54 as
	2,3-diaminopyridine bradykinin B1 receptor antagonists. [My Copy] J Med Chem, Vol. 47, No. 26. (16 December 2004), pp. 6439-6442. by S. D. Kuduk, C. Ng, D. M. Feng, et al.J. M. Wai, R. S. Chang, C. M. Harrell, K. L. Murphy, R. W. Ransom, D. Reiss, M. Ivarsson, G. Mason, S. Boyce, C. Tang, T. Prueksaritanont, R. M. Freidinger, D. J. Pettibone, M. G. Bock posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:34:20 as
	Cyclopropylamino acid amide as a pharmacophoric replacement for 2,3-diaminopyridine. Application to the design of novel bradykinin B1 receptor antagonists. [My Copy] J Med Chem, Vol. 49, No. 4. (23 February 2006), pp. 1231-1234. by M. R. Wood, K. M. Schirripa, J. J. Kim, et al.B. L. Wan, K. L. Murphy, R. W. Ransom, R. S. Chang, C. Tang, T. Prueksaritanont, T. J. Detwiler, L. A. Hettrick, E. R. Landis, Y. M. Leonard, J. A. Krueger, S. D. Lewis, D. J. Pettibone, R. M. Freidinger, M. G. Bock posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:30:27 as
	Potent and orally bioavailable non-peptide antagonists at the human bradykinin B(1) receptor based on a 2-alkylamino-5-sulfamoylbenzamide core. [My Copy] J Med Chem, Vol. 47, No. 19. (9 September 2004), pp. 4642-4644. by T. J. Ritchie, E. K. Dziadulewicz, A. J. Culshaw, et al.W. Müller, G. M. Burgess, G. C. Bloomfield, G. S. Drake, A. R. Dunstan, D. Beattie, G. A. Hughes, P. Ganju, P. McIntyre, S. J. Bevan, C. Davis, M. Yaqoob posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:25:37 as
	New bradykinin analogues modified in the C-terminal part with sterically restricted 1-aminocyclohexane-1-carboxylic acid. [My Copy] J Med Chem, Vol. 48, No. 25. (15 December 2005), pp. 8055-8059. by O. Labudda-Dawidowska, T. H. Wierzba, A. Prahl, et al.W. Kowalczyk, Ł. Gawiński, M. Plackova, J. Slaninová, B. Lammek posted to analogues bradykinin by patricia on 2007-02-22 11:06:11 as
	Structural characterization of cyclic kallidin analogues in DMSO by nuclear magnetic resonance and molecular dynamics. [My Copy] J Pept Sci, Vol. 11, No. 1. (January 2005), pp. 3-16. by E. Schievano, L. Silvestri, M. Gobbo, S. Mammi, R. Rocchi, E. Peggion posted to analogues bioactive bradykinin by patricia on 2007-02-22 10:57:21 as
	Solution-phase combinatorial synthesis of nonpeptide bradykinin antagonists. [My Copy] Bioorg Med Chem, Vol. 12, No. 13. (1 July 2004), pp. 3543-3552. by Y. L. Kam, S. J. Rhee, H. Y. Choo posted to antagonist b2 bradykinin by patricia on 2007-02-22 10:52:32 as
	Spontaneous human B2 bradykinin receptor activity determines the action of partial agonists as agonists or inverse agonists. Effect of basal desensitization. [My Copy] J Biol Chem, Vol. 274, No. 42. (15 October 1999), pp. 29603-29606. by D. B. Fathy, T. Leeb, S. A. Mathis, L. M. Leeb-Lundberg posted to b2 bradykinin mutation receptor by patricia on 2007-02-21 16:38:00 as
	High-affinity binding of peptide agonists to the human B1 bradykinin receptor depends on interaction between the peptide N-terminal L-lysine and the fourth extracellular domain of the receptor. [My Copy] Mol Pharmacol, Vol. 57, No. 1. (January 2000), pp. 171-179. by D. B. Fathy, D. J. Kyle, L. M. Leeb-Lundberg posted to b1 bradykinin mutation receptor by patricia on 2007-02-21 16:33:30 as
	The human B1 bradykinin receptor exhibits high ligand-independent, constitutive activity. Roles of residues in the fourth intracellular and third transmembrane domains. [My Copy] J Biol Chem, Vol. 276, No. 12. (23 March 2001), pp. 8785-8792. by L. M. Leeb-Lundberg, D. S. Kang, M. E. Lamb, D. B. Fathy posted to b1 bradykinin mutation receptor by patricia on 2007-02-21 16:19:26 as
	A single position in the third transmembrane domains of the human B1 and B2 bradykinin receptors is adjacent to and discriminates between the C-terminal residues of subtype-selective ligands. [My Copy] J Biol Chem, Vol. 273, No. 20. (15 May 1998), pp. 12210-12218. by D. B. Fathy, S. A. Mathis, T. Leeb, L. M. Leeb-Lundberg posted to b1 b2 bradykinin mutation receptor by patricia on 2007-02-21 16:00:05 as
	MEN16132, a novel potent and selective nonpeptide antagonist for the human bradykinin B2 receptor. In vitro pharmacology and molecular characterization. [My Copy] Eur J Pharmacol, Vol. 528, No. 1-3. (28 December 2005), pp. 7-16. by P. Cucchi, S. Meini, A. Bressan, et al.C. Catalani, F. Bellucci, P. Santicioli, A. Lecci, A. Faiella, L. Rotondaro, S. Giuliani, A. Giolitti, L. Quartara, C. A. Maggi posted to antagonist b2 bradykinin by patricia on 2007-02-20 17:10:56 as
	The role of helix 8 and of the cytosolic C-termini in the internalization and signal transduction of B(1) and B(2) bradykinin receptors. [My Copy] FEBS J, Vol. 272, No. 1. (January 2005), pp. 129-140. by A. Faussner, A. Bauer, I. Kalatskaya, et al.S. Schüssler, C. Seidl, D. Proud, M. Jochum posted to b1 b2 bradykinin mutation receptor by patricia on 2007-02-20 16:15:48 as
	Binding modes of dihydroquinoxalinones in a homology model of bradykinin receptor 1. [My Copy] Biochem Biophys Res Commun, Vol. 331, No. 1. (27 May 2005), pp. 159-166. by S. N. Ha, P. J. Hey, R. W. Ransom, et al.C. M. Harrell, K. L. Murphy, R. Chang, T. B. Chen, D. S. Su, M. K. Markowitz, M. G. Bock, R. M. Freidinger, F. J. Hess posted to b1 bradykinin model receptor by patricia on 2007-02-20 14:14:40 as
	Identification of the critical residues of bradykinin receptor B1 for interaction with the kinins guided by site-directed mutagenesis and molecular modeling. [My Copy] Biochemistry, Vol. 45, No. 48. (5 December 2006), pp. 14355-14361. by S. N. Ha, P. J. Hey, R. W. Ransom, et al.M. G. Bock, D. S. Su, K. L. Murphy, R. Chang, T. B. Chen, D. Pettibone, J. F. Hess posted to b1 bradykinin mutation receptor by patricia on 2007-02-20 13:53:56 as
	Identification of a Nonpeptidic and Conformationally Restricted Bradykinin B1 Receptor Antagonist with Anti-Inflammatory Activity. [My Copy] J Med Chem, Vol. 50, No. 4. (22 February 2007), pp. 607-610. by Derin C. D'Amico, Toshi Aya, Jason Human, et al.Christopher Fotsch, Jian J. Chen, Kaustav Biswas, Bobby Riahi, Mark H. Norman, Christopher A. Willoughby, Randall Hungate, Paul J. Reider, Gloria Biddlecome, Dianna Lester-Zeiner, Carlo V. Staden, Eileen Johnson, Augustus Kamassah, Leyla Arik, Judy Wang, Vellarkad N. Viswanadhan, Robert D. Groneberg, James Zhan, Hideo Suzuki, Andras Toro, David A. Mareska, David E. Clarke, Darren M. Harvey, Laurence E. Burgess, Ellen R. Laird, Benny Askew, Gordon Ng posted to antagonist b1 bradykinin by patricia on 2007-02-20 13:42:49 as
	Conformational analysis of the highly potent bradykinin antagonist Hoe-140 by means of two different computational methods. [My Copy] J Biomol Struct Dyn, Vol. 15, No. 4. (February 1998), pp. 639-652. by M. Filizola, N. B. Centeno, M. Cartení-Farina, J. J. Perez posted to analogues bioactive bradykinin by patricia on 2007-02-20 13:36:36 as
	Bradykinin receptors and their antagonists. [My Copy] Eur J Pharmacol, Vol. 348, No. 1. (1 May 1998), pp. 1-10. by D. Regoli, S. Nsa Allogho, A. Rizzi, F. J. Gobeil posted to antagonist bradykinin review by patricia on 2007-02-20 11:38:44 as
	Kinin receptors and their antagonists as novel therapeutic agents. [My Copy] Curr Pharm Des, Vol. 7, No. 2. (January 2001), pp. 135-161. by Y. Oztürk posted to antagonist bradykinin review by patricia on 2007-02-20 11:34:01 as
	The potential role of bradykinin antagonists in the treatment of asthma. [My Copy] Agents Actions Suppl, Vol. 38 ( Pt 3) (1992), pp. 439-449. by W. M. Abraham posted to antagonist asthma bradykinin pharmacology by patricia on 2007-02-20 11:26:25 as
	Peptide and non-peptide bradykinin receptor antagonists: role in allergic airway disease. [My Copy] Eur J Pharmacol, Vol. 533, No. 1-3. (8 March 2006), pp. 215-221. by W. M. Abraham, M. Scuri, S. G. Farmer posted to antagonist asthma bradykinin pharmacology review by patricia on 2007-02-20 11:23:42 as
	Non-peptide antagonists for kinin B1 receptors: new insights into their therapeutic potential for the management of inflammation and pain. [My Copy] Trends Pharmacol Sci, Vol. 27, No. 12. (December 2006), pp. 646-651. by M. M. Campos, P. C. Leal, R. A. Yunes, J. B. Calixto posted to antagonist b1 bradykinin review by patricia on 2007-02-20 10:54:31 as
	The kallikrein-kinin system: current and future pharmacological targets. [My Copy] J Pharmacol Sci, Vol. 99, No. 1. (September 2005), pp. 6-38. by M. E. Moreau, N. Garbacki, G. Molinaro, N. J. Brown, F. Marceau, A. Adam posted to antagonist bradykinin review by patricia on 2007-02-20 09:33:37 as
	A new class of bradykinin 1 receptor antagonists containing the piperidine acetic acid tetralin core. [My Copy] Bioorg Med Chem Lett, Vol. 16, No. 8. (15 April 2006), pp. 2071-2075. by C. Fotsch, G. Biddlecome, K. Biswas, et al.J. J. Chen, D. C. D'Amico, R. D. Groneberg, N. B. Han, F. Y. Hsieh, A. Kamassah, G. Kumar, D. Lester-Zeiner, Q. Liu, D. A. Mareska, B. B. Riahi, Y. J. Wang, K. Yang, J. Zhan, J. Zhu, E. Johnson, G. Ng, B. C. Askew posted to antagonist b1 bradykinin by patricia on 2007-02-20 09:26:28 as
	New bradykinin analogues substituted in positions 7 and 8 with sterically restricted 1-aminocyclopentane-1-carboxylic acid. [My Copy] J Pept Sci, Vol. 12, No. 12. (December 2006), pp. 775-779. by O. Labudda, T. Wierzba, D. Sobolewski, et al.W. Kowalczyk, M. Sleszyńska, L. Gawiński, M. Plackova, J. Slaninová, A. Prahl posted to analogues bradykinin by patricia on 2007-02-19 17:19:34 as
	Dual antagonists of the bradykinin B1 and B2 receptors based on a postulated common pharmacophore from existing non-peptide antagonists. [My Copy] Biol Chem, Vol. 387, No. 2. (February 2006), pp. 189-194. by G. Morissette, J. Bouthillier, F. Marceau posted to antagonist b1 b2 bradykinin by patricia on 2007-02-19 15:40:12 as
	Design and synthesis of novel sulfonamide-containing bradykinin hB2 receptor antagonists. 1. Synthesis and SAR of alpha,alpha-dimethylglycine sulfonamides. [My Copy] J Med Chem, Vol. 49, No. 12. (15 June 2006), pp. 3602-3613. by D. Fattori, C. Rossi, C. I. Fincham, et al.M. Berettoni, F. Calvani, F. Catrambone, P. Felicetti, M. Gensini, R. Terracciano, M. Altamura, A. Bressan, S. Giuliani, C. A. Maggi, S. Meini, C. Valenti, L. Quartara posted to antagonist b2 bradykinin by patricia on 2007-02-19 14:32:36 as
	Nonpeptide antagonists for kinin receptors. [My Copy] Regul Pept, Vol. 80, No. 1-2. (17 March 1999), pp. 13-26. by M. Altamura, S. Meini, L. Quartara, C. A. Maggi posted to antagonist bradykinin review by patricia on 2007-02-19 14:24:25 as
	Bradykinin B2 and GPR100 receptors: a paradigm for receptor signal transduction pharmacology [My Copy] Vol. 143, No. 8. (15 November 2004), pp. 938-941. by Stefania Meini, Francesca Bellucci, Paola Cucchi, et al.Sandro Giuliani, Laura Quartara, Alessandro Giolitti, Sabrina Zappitelli, Luigi Rotondaro, Katrin Boels, Carlo A. Maggi posted to bradykinin receptor by patricia on 2007-02-19 14:21:45 as
	Bradykinin antagonists modified with dipeptide mimetic beta-turn inducers. [My Copy] Bioorg Med Chem Lett, Vol. 16, No. 9. (1 May 2006), pp. 2387-2390. by M. C. Alcaro, V. Vinci, A. M. D'Ursi, et al.M. Scrima, M. Chelli, S. Giuliani, S. Meini, M. Di Giacomo, L. Colombo, A. M. Papini posted to analogues bradykinin by patricia on 2007-02-19 14:18:37 as
	Design and synthesis of novel sulfonamide-containing bradykinin hB2 receptor antagonists. 2. Synthesis and structure-activity relationships of alpha,alpha-cycloalkylglycine sulfonamides. [My Copy] J Med Chem, Vol. 50, No. 3. (8 February 2007), pp. 550-565. by D. Fattori, C. Rossi, C. I. Fincham, et al.V. Caciagli, F. Catrambone, P. D'Andrea, P. Felicetti, M. Gensini, E. Marastoni, R. Nannicini, M. Paris, R. Terracciano, A. Bressan, S. Giuliani, C. A. Maggi, S. Meini, C. Valenti, L. Quartara posted to antagonist b2 bradykinin by patricia on 2007-02-19 14:16:34 as
	Bradykinin analogs containing the 4-amino-2-benzazepin-3-one scaffold at the <I>C</I>-terminus [My Copy] Journal of Peptide Science, Vol. 13, No. 3. (2007), pp. 164-170. by S. Ballet, R. De Wachter, K. Van Rompaey, et al. Cs, D. Feytens, G. Töth, L. Quartara, P. Cucchi, S. Meini, D. Tourwé posted to analogues bradykinin by patricia on 2007-02-19 11:11:20 as
	Constitutive activation of the human bradykinin B2 receptor induced by mutations in transmembrane helices III and VI. [My Copy] Mol Pharmacol, Vol. 55, No. 1. (January 1999), pp. 92-101. by J. Marie, C. Koch, D. Pruneau, et al.J. L. Paquet, T. Groblewski, R. Larguier, C. Lombard, B. Deslauriers, B. Maigret, J. C. Bonnafous posted to b2 bradykinin mutation receptor by patricia on 2005-11-30 14:51:00 as
	Mutations in the B2 bradykinin receptor reveal a different pattern of contacts for peptidic agonists and peptidic antagonists. [My Copy] J Biol Chem, Vol. 271, No. 45. (8 November 1996), pp. 28277-28286. by K. Jarnagin, S. Bhakta, P. Zuppan, et al.C. Yee, T. Ho, T. Phan, R. Tahilramani, J. H. Pease, A. Miller, R. Freedman posted to b2 bradykinin mutation receptor by patricia on 2005-11-30 11:18:53 as
	The N terminus of bradykinin when bound to the human bradykinin B2 receptor is adjacent to extracellular Cys20 and Cys277 in the receptor. [My Copy] J Biol Chem, Vol. 271, No. 47. (22 November 1996), pp. 29746-29751. by M. C. Herzig, N. R. Nash, M. Connolly, D. J. Kyle, L. M. Leeb-Lundberg posted to b2 bradykinin mutation receptor by patricia on 2005-11-30 11:10:03 as

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bradykinin	76
antagonist	49
b2	30
receptor	22
b1	17
analogues	15
mutation	15
review	15
gpcr	8
pharmacology	6
bioactive	4
md	3
pharmacophore	3
activation	2
asthma	2
algorithm	1
cancer	1
charges	1
function	1
general	1
inflammation	1
model	1
modeling	1
structure	1

patricia's library 90 articles Export

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