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	Constitutive activation of the alpha 1B-adrenergic receptor by all amino acid substitutions at a single site. Evidence for a region which constrains receptor activation. [My Copy] J Biol Chem, Vol. 267, No. 3. (25 January 1992), pp. 1430-1433. by M. A. Kjelsberg, S. Cotecchia, J. Ostrowski, M. G. Caron, R. J. Lefkowitz posted to activation general gpcr by patricia on 2007-05-14 11:21:34 as
	Coulombic and hydrophobic interactions in the first intracellular loop are vital for bradykinin B2 receptor ligand binding and consequent signal transduction. [My Copy] Biochemistry, Vol. 44, No. 14. (12 April 2005), pp. 5295-5306. by J. Yu, P. Polgar, D. Lubinsky, et al.M. Gupta, L. Wang, D. Mierke, L. Taylor posted to b2 bradykinin mutation receptor by patricia on 2005-11-29 11:26:57 as
	Formulation of 3D pharmacophore models for bradykinin B-2-receptor antagonists [My Copy] LETTERS IN PEPTIDE SCIENCE, Vol. 5, No. 2-3. (May 1998), pp. 189-192. by L. F. Pineda, M. Hassan posted to antagonist b2 bradykinin pharmacophore by patricia on 2005-10-06 16:24:36 as
	Novel non-peptide lead structures for Bradykinin B2-receptor antagonists [My Copy] LETTERS IN PEPTIDE SCIENCE, Vol. 7, No. 2. (March 2000), pp. 69-77. by L. F. Pineda, C. Liebmann, S. Hensellek posted to antagonist b2 bradykinin pharmacophore by patricia on 2005-10-06 16:13:26 as
	International union of pharmacology. XLV. Classification of the kinin receptor family: from molecular mechanisms to pathophysiological consequences. [My Copy] Pharmacol Rev, Vol. 57, No. 1. (March 2005), pp. 27-77. by L. M. Leeb-Lundberg, F. Marceau, W. Müller-Esterl, D. J. Pettibone, B. L. Zuraw posted to antagonist bradykinin receptor review by patricia on 2005-10-04 16:47:06 as
	Site-directed mutagenesis at the human B2 receptor and molecular modelling to define the pharmacophore of non-peptide bradykinin receptor antagonists. [My Copy] Biochem Pharmacol, Vol. 67, No. 4. (15 February 2004), pp. 601-609. by S. Meini, P. Cucchi, F. Bellucci, et al.C. Catalani, A. Faiella, L. Rotondaro, L. Quartara, A. Giolitti, C. A. Maggi posted to b2 bradykinin mutation pharmacophore receptor by patricia on 2005-10-04 16:30:27 as
	Bradykinin antagonists: new opportunities. [My Copy] Curr Opin Chem Biol, Vol. 4, No. 4. (August 2000), pp. 401-406. by M. G. Bock, J. Longmore posted to antagonist bradykinin review by patricia on 2005-10-04 16:00:01 as
	Bradykinin antagonists: discovery and development. [My Copy] Peptides, Vol. 25, No. 3. (March 2004), pp. 527-532. by J. M. Stewart posted to antagonist bradykinin review by patricia on 2005-10-04 15:35:37 as
	Bradykinin receptor ligands: therapeutic perspectives. [My Copy] Nat Rev Drug Discov, Vol. 3, No. 10. (October 2004), pp. 845-852. by F. Marceau, D. Regoli posted to antagonist bradykinin review by patricia on 2005-10-04 15:28:19 as
	Effect of different treatments of long-range interactions and sampling conditions in molecular dynamic simulations of rhodopsin embedded in a dipalmitoyl phosphatidylcholine bilayer. [My Copy] J Comput Chem (31 January 2007) by Arnau Cordomí, Olle Edholm, Juan J J. Perez posted to gpcr receptor by patricia on 2007-03-02 12:24:05 as along with 2 people and 1 group xdeupi arnaucordomi LabCompMed
	Critical role of electrostatic interactions of amino acids at the cytoplasmic region of helices 3 and 6 in rhodopsin conformational properties and activation. [My Copy] J Biol Chem (23 February 2007) by Eva Ramon, Arnau Cordomi, Laia Bosch, et al.Evgeni Yu Y. Zernii, Ivan I I. Senin, Joan Manyosa, Pavel P P. Philippov, Juan J J. Perez, Pere Garriga posted to gpcr receptor by patricia on 2007-03-02 12:02:14 as along with 1 person arnaucordomi
	Dual antagonists of the bradykinin B1 and B2 receptors based on a postulated common pharmacophore from existing non-peptide antagonists. [My Copy] Biol Chem, Vol. 387, No. 2. (February 2006), pp. 189-194. by G. Morissette, J. Bouthillier, F. Marceau posted to antagonist b1 b2 bradykinin by patricia on 2007-02-19 15:40:12 as
	Bradykinin analogs containing the 4-amino-2-benzazepin-3-one scaffold at the <I>C</I>-terminus [My Copy] Journal of Peptide Science, Vol. 13, No. 3. (2007), pp. 164-170. by S. Ballet, R. De Wachter, K. Van Rompaey, et al. Cs, D. Feytens, G. Töth, L. Quartara, P. Cucchi, S. Meini, D. Tourwé posted to analogues bradykinin by patricia on 2007-02-19 11:11:20 as
	Constitutive activation of the human bradykinin B2 receptor induced by mutations in transmembrane helices III and VI. [My Copy] Mol Pharmacol, Vol. 55, No. 1. (January 1999), pp. 92-101. by J. Marie, C. Koch, D. Pruneau, et al.J. L. Paquet, T. Groblewski, R. Larguier, C. Lombard, B. Deslauriers, B. Maigret, J. C. Bonnafous posted to b2 bradykinin mutation receptor by patricia on 2005-11-30 14:51:00 as
	Preliminary mutational analysis of the human kinin B2 receptor for nonpeptide antagonist ligands recognition. [My Copy] Can J Physiol Pharmacol, Vol. 80, No. 4. (April 2002), pp. 303-309. by S. Meini, P. Cucchi, S. Zappitelli, et al.L. Rotondaro, L. Quartara, A. Giolitti, C. A. Maggi posted to antagonist b2 bradykinin mutation receptor by patricia on 2005-11-30 10:47:06 as
	Design and synthesis of novel pyrrolidine-containing bradykinin antagonists. [My Copy] Bioorg Med Chem Lett, Vol. 13, No. 11. (2 June 2003), pp. 1879-1882. by J. Lee, C. Reynolds, M. C. Jetter, et al.M. A. Youngman, D. J. Hlasta, S. L. Dax, D. J. Stone, S. P. Zhang, E. E. Codd posted to antagonist b2 bradykinin by patricia on 2005-11-29 11:33:14 as
	A comparative NMR and molecular dynamics study of the conformations of bradykinin B1 and B2, B2, and B1-specific receptor antagonists B-9430, B-9436, and B-9858. [My Copy] Biopolymers, Vol. 42, No. 5. (15 October 1997), pp. 521-535. by J. Sejbal, Y. Wang, J. R. Cann, J. M. Stewart, L. Gera, G. Kotovych posted to analogues bradykinin by patricia on 2005-11-29 11:31:22 as
	New conformationally homogeneous beta-turn antagonists of the human B2 kinin receptor. [My Copy] J Pept Sci, Vol. 7, No. 5. (May 2001), pp. 270-283. by E. S. Monteagudo, F. Calvani, F. Catrambone, et al.C. I. Fincham, A. Madami, S. Meini, R. Terracciano posted to analogues bradykinin by patricia on 2005-10-04 16:32:03 as
	Non-peptide antagonists and agonists of the bradykinin B(2) receptor. [My Copy] Curr Med Chem, Vol. 9, No. 9. (May 2002), pp. 913-928. by H. Heitsch posted to antagonist bradykinin review by patricia on 2005-10-04 16:24:52 as
	Orphan G-protein-coupled receptors: the next generation of drug targets? [My Copy] Br J Pharmacol, Vol. 125, No. 7. (December 1998), pp. 1387-1392. by S. Wilson, D. J. Bergsma, J. K. Chambers, et al.A. I. Muir, K. G. Fantom, C. Ellis, P. R. Murdock, N. C. Herrity, J. M. Stadel posted to gpcr review by patricia on 2005-10-04 16:17:09 as
	Potent bradykinin antagonists containing N-benzylglycine or N-benzyl-l-alanine in position 8. [My Copy] J Pept Res, Vol. 63, No. 1. (January 2004), pp. 29-35. by O. Dawidowska, A. Prahl, W. Kowalczyk, et al.I. Derdowska, B. Lammek, T. H. Wierzba, W. Juzwa, K. Neubert, J. Zabrocki, B. Olejniczak posted to analogues bradykinin by patricia on 2005-10-04 16:09:36 as
	Conformation mining: an algorithm for finding biologically relevant conformations. [My Copy] J Med Chem, Vol. 48, No. 9. (5 May 2005), pp. 3313-3318. by S. Putta, G. A. Landrum, J. E. Penzotti posted to algorithm bioactive md by patricia on 2005-10-04 16:04:09 as
	Nonpeptide bradykinin B2 receptor antagonists: conversion of rodent-selective bradyzide analogues into potent, orally-active human bradykinin B2 receptor antagonists. [My Copy] J Med Chem, Vol. 45, No. 11. (23 May 2002), pp. 2160-2172. by E. K. Dziadulewicz, T. J. Ritchie, A. Hallett, et al.C. R. Snell, J. W. Davies, R. Wrigglesworth, A. R. Dunstan, G. C. Bloomfield, G. S. Drake, P. McIntyre, M. C. Brown, G. M. Burgess, W. Lee, C. Davis, M. Yaqoob, S. B. Phagoo, E. Phillips, M. N. Perkins, E. A. Campbell, A. J. Davis, H. P. Rang posted to antagonist b2 bradykinin by patricia on 2005-10-04 16:02:22 as
	Bradyzide, a potent non-peptide B(2) bradykinin receptor antagonist with long-lasting oral activity in animal models of inflammatory hyperalgesia. [My Copy] Br J Pharmacol, Vol. 129, No. 1. (January 2000), pp. 77-86. by G. M. Burgess, M. N. Perkins, H. P. Rang, et al.E. A. Campbell, M. C. Brown, P. McIntyre, L. Urban, E. K. Dziadulewicz, T. J. Ritchie, A. Hallett, C. R. Snell, R. Wrigglesworth, W. Lee, C. Davis, S. B. Phagoo, A. J. Davis, E. Phillips, G. S. Drake, G. A. Hughes, A. Dunstan, G. C. Bloomfield posted to antagonist b2 bradykinin by patricia on 2005-10-04 16:01:32 as
	Discovery of orally active nonpeptide bradykinin B2 receptor antagonists. [My Copy] Immunopharmacology, Vol. 43, No. 2-3. (September 1999), pp. 163-168. by M. Asano, N. Inamura, C. Hatori, et al.H. Sawai, T. Fujiwara, Y. Abe, H. Kayakiri, S. Satoh, T. Oku, K. Nakahara posted to antagonist b2 bradykinin by patricia on 2005-10-04 15:53:07 as
	New insights into the conformational requirements of B2 bradykinin antagonism. [My Copy] Bioorg Med Chem, Vol. 6, No. 9. (September 1998), pp. 1491-1500. by M. Filizola, O. Llorens, M. Cartení-Farina, J. J. Perez posted to analogues bioactive bradykinin by patricia on 2005-10-04 15:47:53 as
	A non-peptide antagonist unusually selective for the human form of the bradykinin B2 receptor. [My Copy] Int Immunopharmacol, Vol. 3, No. 10-11. (October 2003), pp. 1529-1536. by F. Marceau, J. P. Fortin, G. Morissette, E. K. Dziadulewicz posted to antagonist b2 bradykinin by patricia on 2005-10-04 15:29:34 as
	A new series of highly potent non-peptide bradykinin B2 receptor antagonists incorporating the 4-heteroarylquinoline framework. Improvement of aqueous solubility and new insights into species difference. [My Copy] J Med Chem, Vol. 47, No. 7. (25 March 2004), pp. 1617-1630. by Y. Sawada, H. Kayakiri, Y. Abe, et al.K. Imai, T. Mizutani, N. Inamura, M. Asano, I. Aramori, C. Hatori, A. Katayama, T. Oku, H. Tanaka posted to antagonist bradykinin by patricia on 2005-10-04 15:21:06 as
	Discovery of the first non-peptide full agonists for the human bradykinin B(2) receptor incorporating 4-(2-picolyloxy)quinoline and 1-(2-picolyl)benzimidazole frameworks. [My Copy] J Med Chem, Vol. 47, No. 11. (20 May 2004), pp. 2853-2863. by Y. Sawada, H. Kayakiri, Y. Abe, et al.T. Mizutani, N. Inamura, M. Asano, C. Hatori, I. Aramori, T. Oku, H. Tanaka posted to antagonist bradykinin by patricia on 2005-10-04 15:20:29 as
	Bradykinin receptor antagonists. [My Copy] IDrugs, Vol. 2, No. 6. (June 1999), pp. 567-575. by H. Heitsch posted to antagonist bradykinin by patricia on 2005-10-04 15:01:26 as
	A novel class of orally active non-peptide bradykinin B2 receptor antagonists. 3. Discovering bioisosteres of the imidazo[1,2-a] pyridine moiety. [My Copy] J Med Chem, Vol. 41, No. 21. (8 October 1998), pp. 4062-4079. by Y. Abe, H. Kayakiri, S. Satoh, et al.T. Inoue, Y. Sawada, N. Inamura, M. Asano, I. Aramori, C. Hatori, H. Sawai, T. Oku, H. Tanaka posted to antagonist bradykinin by patricia on 2005-10-04 14:53:12 as
	A new class of nonpeptide bradykinin B(2) receptor ligand, incorporating a 4-aminoquinoline framework. Identification of a key pharmacophore to determine species difference and agonist/antagonist profile. [My Copy] J Med Chem, Vol. 47, No. 10. (6 May 2004), pp. 2667-2677. by Y. Sawada, H. Kayakiri, Y. Abe, et al.T. Mizutani, N. Inamura, M. Asano, I. Aramori, C. Hatori, T. Oku, H. Tanaka posted to antagonist b2 bradykinin by patricia on 2005-10-04 14:44:21 as
	The structure and function of G-protein-coupled receptors [My Copy] Nature, Vol. 459, No. 7245. (20 May 2009), pp. 356-363. by Daniel M. Rosenbaum, Soren G. F. Rasmussen, Brian K. Kobilka posted to function gpcr review structure by patricia on 2009-06-10 17:23:25 as along with 8 people diod guhjy viktor21614 agrossfield xdeupi akundaje hsekiguc barry
	Nonallergic angioedema: role of bradykinin [My Copy] Allergy, Vol. 62, No. 8. (August 2007), pp. 842-856. by Bas, M., Adams, et al. V., Suvorava, T., Niehues, T., Hoffmann, T. K., Kojda, G. posted to bradykinin pharmacology by patricia on 2007-08-31 09:42:58 as
	B-9972 is an inactivation-resistant agonist of the bradykinin B2 receptor derived from the peptide antagonist B-9430: pharmacologic profile and effective induction of receptor degradation. [My Copy] J Pharmacol Exp Ther (15 August 2007) by Marie-Therese T. Bawolak, Lajos Gera, Guillaume Morissette, John M M. Stewart, Francois Marceau posted to analogues b2 by patricia on 2007-08-31 09:28:14 as
	Novel series of O-substituted 8-quinolines and 4-benzothiazoles as potent antagonists of the bradykinin B2 receptors. [My Copy] Bioorg Med Chem Lett, Vol. 9, No. 3. (8 February 1999), pp. 327-332. by H. Heitsch, A. Wagner, B. A. Schölkens, K. Wirth posted to antagonist b2 bradykinin by patricia on 2007-03-14 12:14:30 as
	Bradykinin B2 receptor as a potential therapeutic target. [My Copy] Drug News Perspect, Vol. 13, No. 4. (May 2000), pp. 213-225. by H. Heitsch posted to b2 pharmacology receptor by patricia on 2007-03-14 12:11:59 as
	Na+ ions binding to the bradykinin B2 receptor suppress agonist-independent receptor activation. [My Copy] Biochemistry, Vol. 35, No. 41. (15 October 1996), pp. 13368-13377. by U. Quitterer, S. AbdAlla, K. Jarnagin, W. Müller-Esterl posted to b2 bradykinin mutation receptor by patricia on 2007-03-02 15:45:35 as
	Identification of a ligand-dependent switch within a muscarinic receptor. [My Copy] J Biol Chem, Vol. 273, No. 34. (21 August 1998), pp. 21563-21568. by T. A. Spalding, E. S. Burstein, S. C. Henderson, K. R. Ducote, M. R. Brann posted to activation gpcr receptor by patricia on 2007-03-02 13:20:40 as
	Biomolecular modeling: Goals, problems, perspectives. [My Copy] Angewandte Chemie (International ed. in English), Vol. 45, No. 25. (19 June 2006), pp. 4064-4092. by Wilfred F. van Gunsteren, Dirk Bakowies, Riccardo Baron, et al.Indira Chandrasekhar, Markus Christen, Xavier Daura, Peter Gee, Daan P. Geerke, Alice Glättli, Philippe H. Hünenberger, Mika A. Kastenholz, Chris Oostenbrink, Merijn Schenk, Daniel Trzesniak, Nico F. van der Vegt, Haibo B. Yu posted to md modeling review by patricia on 2007-02-23 11:33:08 as along with 2 people mijogiffin LamBras
	G-protein-coupled receptors and cancer [My Copy] Nature Reviews Cancer, Vol. 7, No. 2., pp. 79-94. by Robert T. Dorsam, Silvio J. Gutkind posted to cancer gpcr by patricia on 2007-02-23 09:56:25 as
	Nonpeptide ligands that target peptide-activated GPCRs in inflammation. [My Copy] Curr Med Chem, Vol. 12, No. 25. (2005), pp. 3027-3042. by J. S. Blakeney, D. P. Fairlie posted to antagonist gpcr inflammation by patricia on 2007-02-22 11:52:52 as
	Bradykinin B1 antagonists: SAR studies in the 2,3-diaminopyridine series. [My Copy] Bioorg Med Chem Lett, Vol. 15, No. 17. (1 September 2005), pp. 3925-3929. by S. D. Kuduk, R. K. Chang, C. Ng, et al.K. L. Murphy, R. W. Ransom, C. Tang, T. Prueksaritanont, R. M. Freidinger, D. J. Pettibone, M. G. Bock posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:47:57 as
	2,3-Diaminopyridine as a platform for designing structurally unique nonpeptide bradykinin B1 receptor antagonists. [My Copy] Bioorg Med Chem Lett, Vol. 15, No. 9. (2 May 2005), pp. 2385-2388. by D. M. Feng, J. M. Wai, S. D. Kuduk, et al.C. Ng, K. L. Murphy, R. W. Ransom, D. Reiss, R. S. Chang, C. M. Harrell, T. MacNeil, C. Tang, T. Prueksaritanont, R. M. Freidinger, D. J. Pettibone, M. G. Bock posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:45:05 as
	5-Piperazinyl pyridine carboxamide bradykinin B1 antagonists. [My Copy] Bioorg Med Chem Lett, Vol. 16, No. 10. (15 May 2006), pp. 2791-2795. by S. D. Kuduk, C. N. Di Marco, R. K. Chang, et al.M. R. Wood, J. J. Kim, K. M. Schirripa, K. L. Murphy, R. W. Ransom, C. Tang, M. Torrent, S. Ha, T. Prueksaritanont, D. J. Pettibone, M. G. Bock posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:38:54 as
	2,3-diaminopyridine bradykinin B1 receptor antagonists. [My Copy] J Med Chem, Vol. 47, No. 26. (16 December 2004), pp. 6439-6442. by S. D. Kuduk, C. Ng, D. M. Feng, et al.J. M. Wai, R. S. Chang, C. M. Harrell, K. L. Murphy, R. W. Ransom, D. Reiss, M. Ivarsson, G. Mason, S. Boyce, C. Tang, T. Prueksaritanont, R. M. Freidinger, D. J. Pettibone, M. G. Bock posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:34:20 as
	Cyclopropylamino acid amide as a pharmacophoric replacement for 2,3-diaminopyridine. Application to the design of novel bradykinin B1 receptor antagonists. [My Copy] J Med Chem, Vol. 49, No. 4. (23 February 2006), pp. 1231-1234. by M. R. Wood, K. M. Schirripa, J. J. Kim, et al.B. L. Wan, K. L. Murphy, R. W. Ransom, R. S. Chang, C. Tang, T. Prueksaritanont, T. J. Detwiler, L. A. Hettrick, E. R. Landis, Y. M. Leonard, J. A. Krueger, S. D. Lewis, D. J. Pettibone, R. M. Freidinger, M. G. Bock posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:30:27 as
	Potent and orally bioavailable non-peptide antagonists at the human bradykinin B(1) receptor based on a 2-alkylamino-5-sulfamoylbenzamide core. [My Copy] J Med Chem, Vol. 47, No. 19. (9 September 2004), pp. 4642-4644. by T. J. Ritchie, E. K. Dziadulewicz, A. J. Culshaw, et al.W. Müller, G. M. Burgess, G. C. Bloomfield, G. S. Drake, A. R. Dunstan, D. Beattie, G. A. Hughes, P. Ganju, P. McIntyre, S. J. Bevan, C. Davis, M. Yaqoob posted to antagonist b1 bradykinin by patricia on 2007-02-22 11:25:37 as
	New bradykinin analogues modified in the C-terminal part with sterically restricted 1-aminocyclohexane-1-carboxylic acid. [My Copy] J Med Chem, Vol. 48, No. 25. (15 December 2005), pp. 8055-8059. by O. Labudda-Dawidowska, T. H. Wierzba, A. Prahl, et al.W. Kowalczyk, Ł. Gawiński, M. Plackova, J. Slaninová, B. Lammek posted to analogues bradykinin by patricia on 2007-02-22 11:06:11 as
	Structural characterization of cyclic kallidin analogues in DMSO by nuclear magnetic resonance and molecular dynamics. [My Copy] J Pept Sci, Vol. 11, No. 1. (January 2005), pp. 3-16. by E. Schievano, L. Silvestri, M. Gobbo, S. Mammi, R. Rocchi, E. Peggion posted to analogues bioactive bradykinin by patricia on 2007-02-22 10:57:21 as

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