xdeupi's pharmacology [31 articles] Export

Recent papers added to xdeupi's library classified by the tag pharmacology. You can also see everyone's pharmacology.

	The impact of GPCR structures on pharmacology and structure-based drug design. [My Copy] British journal of pharmacology (13 November 2009) by Miles Congreve, Fiona Marshall posted to review pharmacology gpcr by xdeupi on 2009-11-20 12:39:25 as
	Web Server To Identify Similarity of Amino Acid Motifs to Compounds (SAAMCO) [My Copy] Journal of Chemical Information and Modeling, Vol. 48, No. 7. (1 July 2008), pp. 1524-1529. by Fergal P. Casey, Norman E. Davey, Ivan Baran, Radka S. Varekova, Denis C. Shields posted to webserver theory pharmacology ligands drug by xdeupi on 2009-10-05 18:46:59 as along with 1 person higueruelo
	Hot-Spots-Guided Receptor-Based Pharmacophores (HS-Pharm): A Knowledge-Based Approach to Identify Ligand-Anchoring Atoms in Protein Cavities and Prioritize Structure-Based Pharmacophores [My Copy] Journal of Chemical Information and Modeling, Vol. 48, No. 7. (1 July 2008), pp. 1396-1410. by Caterina Barillari, Gilles Marcou, Didier Rognan posted to theory pharmacology ligands drug docking binding b2ar agonist by xdeupi on 2009-10-05 18:45:05 as along with 3 people tbinbal superpyrin higueruelo
	Allosteric modulation of muscarinic acetylcholine receptors. [My Copy] Current neuropharmacology, Vol. 5, No. 3. (September 2007), pp. 157-167. by K. J. Gregory, P. M. Sexton, A. Christopoulos posted to activation agonist binding kinetics ligands pharmacology by xdeupi on 2009-07-20 18:21:37 as
	Validity of (−)-[<sup>3</sup>H]-CGP 12177A as a radioligand for the 'putative <i>β</i><sub>4</sub>-adrenoceptor' in rat atrium [My Copy] British Journal of Pharmacology, Vol. 123, No. 3. (1998), pp. 371-380. by Doreen Sarsero, Peter Molenaar, Alberto J. Kaumann posted to b1ar ligands pharmacology by xdeupi on 2009-06-10 13:56:13 as
	Sequence-Derived Three-Dimensional Pharmacophore Models for G-Protein-Coupled Receptors and Their Application in Virtual Screening [My Copy] Journal of Medicinal Chemistry, Vol. 0, No. 0. (0000) by Thomas Klabunde, Clemens Giegerich, Andreas Evers posted to agonist antagonist binding drug ligands modeling pharmacology by xdeupi on 2009-05-06 09:59:59 as along with 1 person reyez
	Physiological relevance of GPCR oligomerization and its impact on drug discovery. [My Copy] Drug discovery today, Vol. 13, No. 23-24. (14 December 2008), pp. 1059-1066. by Rosemarie Panetta, Michael T. Greenwood posted to dimer disease drug gpcr ligands pharmacology review by xdeupi on 2008-10-16 09:57:50 as along with 1 person guhjy
	Recruitment of beta-arrestin2 to the dopamine D2 receptor: Insights into anti-psychotic and anti-parkinsonian drug receptor signaling. [My Copy] Neuropharmacology (8 April 2008) by Ib V V. Klewe, Søren M M. Nielsen, Louise Tarpø, et al.Eneko Urizar, Concetta Dipace, Jonathan A A. Javitch, Ulrik Gether, Jan Egebjerg, Kenneth V V. Christensen posted to activation active-state agonist arrestin biased_agonism binding disease fluorescence imaging internalization pharmacology by xdeupi on 2008-05-13 16:24:49 as
	Clinical consequences of ADR2 polymorphisms [My Copy] Pharmacogenomics, Vol. 9, No. 3. (March 2008), pp. 349-358. by Hawkins, A. Gregory, Weiss, T. Scott, Bleecker, R. Eugene posted to b2ar disease drug genome pharmacology polymorphism review by xdeupi on 2008-05-03 17:12:39 as
	Functional assays as prismatic views of drug activity: relevance to new drug discovery. [My Copy] Journal of receptor and signal transduction research, Vol. 28, No. 1. (2008), pp. 109-125. by T. Kenakin posted to biased_agonism chemokine drug pharmacology review by xdeupi on 2008-05-03 17:03:08 as
	Chemogenomic approaches to rational drug design [My Copy] Br J Pharmacol, Vol. 152, No. 1. (29 May 2007), pp. 38-52. by D. Rognan posted to agonist binding drug ligands pharmacology priviledged_structures by xdeupi on 2008-03-28 15:54:47 as along with 4 people and 3 groups jmrivort jerome_ucsf_slb guhjy tjimenez LabCompMed G-quadruplex Supramolecular
	beta-Arrestin-biased Agonism at the beta2-Adrenergic Receptor. [My Copy] J Biol Chem, Vol. 283, No. 9. (29 February 2008), pp. 5669-5676. by M. T. Drake, J. D. Violin, E. J. Whalen, J. W. Wisler, S. K. Shenoy, R. J. Lefkowitz posted to activation agonist arrestin b2ar biased_agonism drug gproteins imaging internalization ligands pharmacology by xdeupi on 2008-02-27 10:39:07 as along with 1 group LabCompMed
	G-protein-coupled receptor signalling through protein networks. [My Copy] Biochem Soc Trans, Vol. 35, No. Pt 1. (February 2007), pp. 23-27. by A. D. Strosberg, C. Nahmias posted to b2ar gpcr pharmacology review structure by xdeupi on 2007-06-29 21:10:57 as along with 1 group LabCompMed
	Heterologous Expression of the Adenosine A1 Receptor in Transgenic Mouse Retina. [My Copy] Biochemistry (20 June 2007) by Ning Li, David Salom, Li Zhang, et al.Tim Harris, Juan A. Ballesteros, Marcin Golczak, Beata Jastrzebska, Krzysztof Palczewski, Carole Kurahara, Todd Juan, Steven Jordan, John A. Salon posted to expression gpcr pharmacology by xdeupi on 2007-06-25 10:09:54 as along with 1 group LabCompMed
	Multiple signaling states of G-protein-coupled receptors. [My Copy] Pharmacol Rev, Vol. 57, No. 2. (June 2005), pp. 147-161. by D. M. Perez, S. S. Karnik posted to activation agonist gpcr pharmacology review rhodopsin switch by xdeupi on 2007-04-26 14:57:25 as along with 1 group LabCompMed
	Smart drug discovery leveraging innovative technologies and predictive knowledge. [My Copy] Nat Chem Biol, Vol. 2, No. 12. (December 2006), pp. 646-648. by T. K. Sawyer posted to drug pharmacology by xdeupi on 2007-04-23 16:56:56 as along with 1 group LabCompMed
	Chemical Biology & Drug Design: First Anniversary - 2007! [My Copy] Chem Biol Drug Des, Vol. 69, No. 1. (January 2007), pp. 1-2. by Tomi K K. Sawyer posted to drug pharmacology review by xdeupi on 2007-04-23 16:56:17 as along with 1 group LabCompMed
	"Phenotypic" pharmacology: the influence of cellular environment on G protein-coupled receptor antagonist and inverse agonist pharmacology. [My Copy] Biochem Pharmacol, Vol. 73, No. 6. (15 March 2007), pp. 737-751. by C. P. Nelson, R. A. Challiss posted to agonist gpcr ligands pharmacology by xdeupi on 2007-04-10 18:54:26 as along with 1 person and 2 groups Fritz neurolit LabCompMed
	Dosage-dependent switch from G protein-coupled to G protein-independent signaling by a GPCR. [My Copy] The EMBO journal, Vol. 26, No. 1. (10 January 2007), pp. 53-64. by Yutong Sun, Jianyun Huang, Yang Xiang, et al.Murat Bastepe, Harald Jüppner, Brian K. Kobilka, Jillian J. Zhang, Xin-Yun Y. Huang posted to activation b2ar drug pharmacology switch by xdeupi on 2007-03-21 11:13:23 as along with 2 people and 1 group diod Guff32 LabCompMed
	Subclassification and nomenclature of alpha- and beta-adrenoceptors. [My Copy] Curr Top Med Chem, Vol. 7, No. 2. (2007), pp. 129-134. by J. P. Hieble posted to agonist b2ar drug genome ligands pharmacology review by xdeupi on 2007-03-12 14:33:19 as along with 1 group LabCompMed
	Recent advances in identification and characterization of beta-adrenoceptor agonists and antagonists. [My Copy] Curr Top Med Chem, Vol. 7, No. 2. (2007), pp. 207-216. by J. P. Hieble posted to agonist b2ar drug ligands pharmacology by xdeupi on 2007-03-12 14:32:04 as along with 1 group LabCompMed
	Both Ligand- and Cell-Specific Parameters Control Ligand Agonism in a Kinetic Model of G Protein-Coupled Receptor Signaling. [My Copy] PLoS Comput Biol, Vol. 3, No. 1. (12 January 2007) by Tamara L L. Kinzer-Ursem, Jennifer J J. Linderman posted to activation agonist b2ar pharmacology by xdeupi on 2007-02-13 15:38:17 as along with 1 group LabCompMed
	I want a new drug: G-protein-coupled receptors in drug development. [My Copy] Drug Discov Today, Vol. 11, No. 11-12. (June 2006), pp. 481-493. by S. Schlyer, R. Horuk posted to cancer drug gpcr ligands pharmacology review by xdeupi on 2006-11-04 12:41:53 as along with 1 person and 1 group zimbo1 LabCompMed
	dummy [My Copy] by Dummy posted to 5ht1a activation agonist amber amine arrestin b2ar bimane binding cam ccr5 channel chemokine chimera crystallography cterm cxcr1 d250 dimer disease drug dry dynamics ecl2 evolution expression fluorescence folding fret genome gly gpcr gproteins hbond helix helix8 histamine hormone icl3 imaging internalization ionic leukotriene lhr ligands lipids lock loops md membrane modeling mutation n745 n749 nmr npxxy nterm opioid pharmacology polymorphism pro-kink protonation review rhodopsin s542 sequence ser spin_labeling structure switch thr thyrotropin tm2 tm3 tm5 tm6 tm7 toggle transmembrane trp txp w648 by xdeupi on 2006-10-30 12:30:16 as along with 2 people and 1 group jessicaopacic ivanrt LabCompMed
	Modeling and active site refinement for G protein-coupled receptors: application to the beta-2 adrenergic receptor. [My Copy] J Comput Aided Mol Des (13 October 2006) by Stanley R. Krystek, S R. Kimura, Andrew J. Tebben posted to b2ar binding drug ligands modeling pharmacology by xdeupi on 2006-10-27 09:43:03 as along with 1 person and 1 group daevans LabCompMed
	Functional selectivity and classical concepts of quantitative pharmacology. [My Copy] J Pharmacol Exp Ther (27 June 2006) by Jonathan D D. Urban, William P P. Clarke, Mark von Zastrow, et al.David E E. Nichols, Brian K K. Kobilka, Harel Weinstein, Jonathan A A. Javitch, Bryan L L. Roth, Arthur Christopoulos, Patrick Sexton, Keith Miller, Michael Spedding, Richard B B. Mailman posted to activation b2ar pharmacology review switch by xdeupi on 2006-09-07 15:43:50 as along with 2 people and 1 group shoshin kentsis LabCompMed
	Novel mutants of the human beta1-adrenergic receptor reveal amino acids relevant for receptor activation. [My Copy] J Biol Chem, Vol. 281, No. 26. (30 June 2006), pp. 18120-18125. by B. Behr, C. Hoffmann, G. Ottolina, K. N. Klotz posted to activation agonist b2ar binding drug ligands modeling mutation pharmacology structure by xdeupi on 2006-09-05 11:05:20 as along with 1 group LabCompMed
	G proteins in drug screening: from analysis of receptor-G protein specificity to manipulation of GPCR-mediated signalling pathways. [My Copy] Curr Pharm Des, Vol. 12, No. 14. (2006), pp. 1703-1715. by E. Kostenis posted to activation cterm drug ecl2 gpcr gproteins pharmacology by xdeupi on 2006-09-05 09:59:05 as along with 1 group LabCompMed
	Determining the Potency and Molecular Mechanism of Action of Insurmountable Antagonists. [My Copy] J Pharmacol Exp Ther (20 July 2006) by Terry P P. Kenakin, Stephen Jenkinson, Christian Watson posted to activation drug ligands agonist pharmacology by xdeupi on 2006-09-05 09:51:58 as along with 1 group LabCompMed
	GPCR agonists and antagonists in the clinic. [My Copy] Med Chem, Vol. 1, No. 4. (July 2005), pp. 405-421. by J. D. Tyndall, R. Sandilya posted to agonist drug gpcr ligands pharmacology by xdeupi on 2006-07-24 10:18:01 as along with 1 group LabCompMed
	Data-Driven Analysis in Drug Discovery [My Copy] Journal of Receptors and Signal Transduction, Vol. 26, No. 4. (August 2006), pp. 299-327. by Terry Kenakin posted to agonist binding drug ligands pharmacology by xdeupi on 2006-07-17 16:28:05 as along with 1 group LabCompMed

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activation	173
gpcr	112
structure	89
rhodopsin	79
review	65
modeling	62
b2ar	58
dynamics	56
helix	50
transmembrane	47
agonist	46
binding	45
theory	44
ligands	41
drug	36
md	35
switch	34
membrane_proteins	31
pharmacology	31
crystallography	30
nmr	30
membrane	26
gproteins	24
dimer	20
fluorescence	18
sequence	17
ser	17
active-state	15
pro-kink	15
folding	14
fret	14
genome	14
loops	14
flexibility	13
disease	12
tm6	12
cterm	11
mutation	11
retinal	11
amber	10
energy_landscape	10
evolution	10
toggle	10
arrestin	9
docking	9
kinetics	9
lipids	9
neurokinin	9
tm5	9
chemokine	8
gpcrs	8
hbond	8
helix8	8
imaging	8
bimane	7
cancer	7
channel	7
ecl2	7
gly	7
icl3	7
ionic	7
lmc_101	7
plasticity	7
protonation	7
tm3	7
w648	7
cation-pi	6
ccr5	6
conformational_changes	6
cys_scanning	6
d250	6
internalization	6
npxxy	6
opioid	6
thyrotropin	6
tm2	6
xray	6
amine	5
binding_kinetics	5
dimerization	5
dry	5
expression	5
lock	5
polymorphism	5
spectroscopy	5
thr	5
trp	5
angiotensin	4
antagonist	4
biased_agonism	4
cam	4
cholesterol	4
disorder	4
hormone	4
n749	4
nterm	4
pathway	4
tm7	4
water	4
cxcr1	3
grk	3
histamine	3
n745	3
oligomerization	3
spin_labeling	3
toac	3
webserver	3
5ht1a	2
chimera	2
crosslinking	2
em	2
leukotriene	2
lhr	2
networks	2
pathways	2
phylogeny	2
s542	2
solvation	2
tm1	2
tmhs	2
txp	2
b1ar	1
binding_site	1
class_c	1
efficacy	1
gaba	1
induced_fit	1
inverse_agonist	1
kinase	1
kinks	1
metai	1
oligomers	1
peptide	1
priviledged_structures	1
protein_docking	1
selectivity	1
sequence_alignment	1
tm4	1
transducin	1
vasopressin	1

xdeupi's pharmacology [31 articles] Export

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